SCHEMBL28053334

SCHEMBL28053334

COc1ncc(S(N)(=O)=O)cc1-c1ccc(Cl)nc1O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.35
CA1 P00915 3/20 0.34
CA2 P00918 3/20 0.34
LRRK2 Q5S007 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
PTGES2 Q9H7Z7 3/20 0.34
SCN9A Q15858 2/20 0.34
BRD4 O60885 1/20 0.34
CA12 O43570 2/20 0.33
CA9 Q16790 2/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
APLNR P35414 1/20 0.33
FYN P06241 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
TDP2 O95551 1/20 0.33
NSD2 O96028 1/20 0.33
GCK P35557 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053340 0.80 PTGS1 (0.42) CA1CA2PTGES2SCN9ABRD4
SCHEMBL28053341 0.77 PKM (0.49) CA1CA2ALDH1A1PKMCA12
SCHEMBL28826183 0.77 APLNR (0.40) CA1CA2PTGES2BRD4CA12
SCHEMBL28053271 0.74 PTGS2 (0.37) CA1CA2ALDH1A1BRD4APLNR
SCHEMBL16235251 0.70 S100A9 (0.58) LRRK2ALDH1A1PTGES2LMNAMAPK1
SCHEMBL28053239 0.65 APLNR (0.38) CA1CA2ALDH1A1BRD4CA12
SCHEMBL28053335 0.65 CA2 (0.42) IKBKBCA1CA2PKMCA12
SCHEMBL1700491 0.64 CA2 (0.39) CA1CA2ALDH1A1PTGES2CA12
SCHEMBL15211939 0.64 PTGES2 (0.45) CA1CA2PTGES2SCN9ACA12
SCHEMBL11335088 0.64 PTGS2 (0.42) CA1CA2PKMCA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN claimed
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN disclosed