SCHEMBL28053341

SCHEMBL28053341

NS(=O)(=O)c1ccc(-c2ccc(Cl)nc2O)c(-c2ccc(Cl)nc2O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 3/20 0.49
POLB P06746 1/20 0.49
GAA P10253 2/20 0.45
MAPT P10636 2/20 0.45
ALDH1A1 P00352 1/20 0.45
TDP2 O95551 1/20 0.45
NSD2 O96028 1/20 0.45
HK1 P19367 1/20 0.45
PAX8 Q06710 1/20 0.45
CA1 P00915 10/20 0.42
CA2 P00918 9/20 0.42
CA9 Q16790 9/20 0.42
CA12 O43570 6/20 0.42
CA7 P43166 3/20 0.41
CA14 Q9ULX7 3/20 0.41
CA4 P22748 2/20 0.41
CA6 P23280 2/20 0.41
CA5A P35218 2/20 0.41
CA5B Q9Y2D0 2/20 0.41
CA3 P07451 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053334 0.77 IKBKB (0.35) PKMALDH1A1TDP2NSD2CA1
SCHEMBL28053258 0.73 PKM (0.46) PKMPOLBGAAMAPTALDH1A1
SCHEMBL29902406 0.69 PKM (0.62) PKMPOLBGAAMAPTALDH1A1
SCHEMBL8349082 0.66 LMNA (0.67) PKMPOLBGAAMAPTALDH1A1
SCHEMBL11117720 0.66 CA2 (0.59) PKMGAAMAPTALDH1A1CA1
SCHEMBL1803937 0.66 PTGS1 (0.66) PKMGAAMAPTCA1CA2
SCHEMBL4709444 0.66 TDP1 (0.60) PKMPOLBGAAMAPTCA1
SCHEMBL10775524 0.66 TDP2 (0.67) PKMPOLBGAAMAPTALDH1A1
SCHEMBL7339146 0.66 TDP2 (0.67) PKMPOLBGAAMAPTALDH1A1
SCHEMBL27954272 0.65 PKM (0.51) PKMPOLBGAAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN claimed
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN disclosed