SCHEMBL28061589

SCHEMBL28061589

FC(F)(F)Oc1c[c]ccc1CC1(CN2CCCC2)CC1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 8/20 0.35
DRD2 P14416 4/20 0.35
SLC6A2 P23975 1/20 0.33
CYP2D6 P10635 1/20 0.33
SLC6A4 P31645 4/20 0.32
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28061573 0.90 ALDH1A1 (0.41) SLC6A3DRD2SLC6A2SLC6A4LMNA
SCHEMBL28061570 0.90 EPHX2 (0.33)
SCHEMBL28061544 0.81 LMNA (0.39) LMNA
SCHEMBL28061552 0.79 LMNA (0.31) SLC6A3SLC6A2SLC6A4LMNA
SCHEMBL28061564 0.75 LIPE (0.35)
SCHEMBL28001641 0.69 SLC6A4 (0.41) SLC6A3SLC6A2CYP2D6SLC6A4LMNA
SCHEMBL3542512 0.68 EPHX2 (0.32)
SCHEMBL21268313 0.68 EPHX2 (0.32)
SCHEMBL28793420 0.68
SCHEMBL16951433 0.66 CTSS (0.34) SLC6A3DRD2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105693645-B Condensed heterocyclic compouds as ion channel modulators 吉利德科学公司 2018-10-09 CN disclosed
CN-105693645-A FUSED HETEROCYCLIC COMPOUNDS AS SODIUM CHANNEL MODULATORS 吉利德科学公司 2016-06-22 CN disclosed
CN-103649056-B Fused heterocyclic compounds as modulators of ion channels GILEAD SCIENCES, INC. (US) 2016-04-27 CN disclosed