SCHEMBL28061573

SCHEMBL28061573

CN1CCN(CC2(Cc3cc[c]cc3OC(F)(F)F)CC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
SLC6A2 P23975 8/20 0.38
SLC6A4 P31645 3/20 0.38
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35
SLC6A3 Q01959 4/20 0.33
DRD2 P14416 3/20 0.33
HTR6 P50406 2/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
HCN1 O60741 1/20 0.31
ABL1 P00519 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28061589 0.90 SLC6A3 (0.35) SLC6A2SLC6A4SLC6A3DRD2LMNA
SCHEMBL28061570 0.86 EPHX2 (0.33) ABL1
SCHEMBL28061544 0.78 LMNA (0.39) LMNA
SCHEMBL28061552 0.76 LMNA (0.31) SLC6A2SLC6A4SLC6A3LMNA
SCHEMBL28061564 0.72 LIPE (0.35) MEN1KMT2A
SCHEMBL27651774 0.70 DRD2 (0.43) ALDH1A1MEN1KMT2AATMSLC6A3
SCHEMBL3542512 0.68 EPHX2 (0.32)
SCHEMBL28001641 0.67 SLC6A4 (0.41) SLC6A2SLC6A4SLC6A3LMNA
SCHEMBL16951433 0.66 CTSS (0.34) SLC6A2SLC6A3DRD2
SCHEMBL222030 0.66 MEN1 (0.49) ALDH1A1MEN1KMT2ADRD2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105693645-A FUSED HETEROCYCLIC COMPOUNDS AS SODIUM CHANNEL MODULATORS 吉利德科学公司 2016-06-22 CN disclosed
CN-103649056-B Fused heterocyclic compounds as modulators of ion channels GILEAD SCIENCES, INC. (US) 2016-04-27 CN disclosed