SCHEMBL28045730

SCHEMBL28045730

O=COC(Cc1ccccc1)Cc1cc[nH]n1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 8/20 0.37
CTSL P07711 4/20 0.36
CTSB P07858 4/20 0.36
EPHX1 P07099 2/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
CTSH P09668 2/20 0.32
CYP1A2 P05177 2/20 0.32
SRR Q9GZT4 2/20 0.31
ACP3 P15309 1/20 0.31
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
ALPI P09923 1/20 0.30
PKM P14618 1/20 0.30
PTGS1 P23219 1/20 0.30
XIAP P98170 1/20 0.30
SLC7A5 Q01650 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28824696 0.86 ALDH1A1 (0.32) ALDH1A1LMNANPSR1
SCHEMBL28825902 0.83 LDHA (0.40) CYP1A2ALDH1A1
SCHEMBL18085416 0.82 EPHX1 (0.48) CTSKCTSLCTSBEPHX1MEN1
SCHEMBL27977725 0.81 AKR1B1 (0.33) MEN1KMT2AALDH1A1
SCHEMBL28061404 0.78 EPHX1 (0.35) CTSKCTSLCTSBEPHX1MEN1
SCHEMBL28113598 0.78 CTSK (0.34) CTSKCTSLCTSBEPHX1MEN1
SCHEMBL28268882 0.78
SCHEMBL28827075 0.78 GLS (0.32)
SCHEMBL28074772 0.77 CTSK (0.36) CTSKCTSLCTSBEPHX1MEN1
SCHEMBL28113592 0.75 TSHR (0.42) CTSKEPHX1MEN1KMT2ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105121432-A Heterocyclic amides as kinase inhibitors GLAXOSMITHKLINE IP DEV LTD 2015-12-02 CN disclosed