Tipepidine

Tipepidine

SCHEMBL28142103

CCC1(CC)C(=O)CCN=C1O.CN1CCCC(=C(c2cccs2)c2cccs2)C1

nearest known ligand 0.34

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
KMT2A Q03164 3/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 4/20 0.32
KCNH2 Q12809 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LMNA P02545 2/20 0.31
GAA P10253 1/20 0.31
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.31
PDE4D Q08499 1/20 0.31
CACNA2D1 P54289 1/20 0.31
NOS3 P29474 3/20 0.31
NOS1 P29475 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MAPK1 P28482 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tipepidine SCHEMBL13723968 0.82 OPRM1 (0.35) OPRM1OPRD1KMT2AMEN1ALDH1A1
Tipepidine SCHEMBL410090 0.78 NOS3 (0.43) KMT2AMEN1ALDH1A1SMN1; SMN2LMNA
Tipepidine SCHEMBL30827547 0.77 NOS3 (0.42) KMT2AMEN1ALDH1A1SMN1; SMN2LMNA
Tipepidine SCHEMBL11026418 0.72 HPGDS (0.43) KMT2AMEN1ALDH1A1SMN1; SMN2LMNA
Tipepidine SCHEMBL663025 0.69 KDM4E (0.41) KMT2AMEN1ALDH1A1SMN1; SMN2LMNA
SCHEMBL11319505 0.59 KMT2A (0.47) KMT2AMEN1ALDH1A1LMNAGAA
SCHEMBL11352518 0.58 HRH2 (0.45) OPRM1OPRD1KMT2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL11354148 0.58 KMT2A (0.46) KMT2AMEN1ALDH1A1LMNAGAA
SCHEMBL11311454 0.57 ALDH1A1 (0.45) OPRM1OPRD1ALDH1A1SMN1; SMN2GAA
SCHEMBL11356487 0.57 HRH2 (0.44) OPRM1OPRD1KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103717597-B Heterocyclic compounds as kinase inhibitors 原真股份有限公司 2017-07-04 CN disclosed