SCHEMBL28224535

SCHEMBL28224535

CCOC(=O)C(F)c1ccc(O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.52
CA12 O43570 4/20 0.52
CA1 P00915 4/20 0.52
CA2 P00918 4/20 0.52
CA7 P43166 4/20 0.52
CA9 Q16790 4/20 0.52
CA14 Q9ULX7 4/20 0.52
ESR2 Q92731 3/20 0.52
KMT2A Q03164 1/20 0.47
LMNA P02545 2/20 0.44
MAPT P10636 2/20 0.44
CHRM1 P11229 2/20 0.44
SLC6A2 P23975 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
CYP1A2 P05177 1/20 0.44
PGR P06401 1/20 0.44
CHRM2 P08172 1/20 0.44
CYP3A4 P08684 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
AR P10275 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27595607 0.85 MAPT (0.47) KMT2ALMNAMAPTTDP1CYP1A2
SCHEMBL18610656 0.84 MAPT (0.46) KMT2ALMNAMAPTTDP1CYP1A2
SCHEMBL11260308 0.84 LMNA (0.53) CA12CA1CA2CA9KMT2A
SCHEMBL2799224 0.84 CA12 (0.50) CA12CA1CA2CA9LMNA
SCHEMBL7987182 0.84 OPRM1 (0.38) CA12CA1CA2CA9KMT2A
SCHEMBL324209 0.83 MMP8 (0.56) CA12CA1CA2CA9KMT2A
SCHEMBL4290959 0.83 MMP8 (0.56) CA12CA1CA2CA9KMT2A
SCHEMBL2400228 0.83 MMP8 (0.56) CA12CA1CA2CA9KMT2A
SCHEMBL22820555 0.82 PTGS2 (0.51) CA12CA1CA2CA9KMT2A
SCHEMBL27462191 0.82 ALDH1A1 (0.43) ESR1CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108239029-A The preparation of tetrahydroisoquinoliderivatives compound and its salt and medical usage 中国医学科学院药物研究所 2018-07-03 CN disclosed