SCHEMBL28293160

SCHEMBL28293160

CC(OC=O)c1c[nH]c2cccc(NS(C)(=O)=O)c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.40
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
NR3C1 P04150 6/20 0.37
PGR P06401 5/20 0.37
NR3C2 P08235 5/20 0.37
AR P10275 5/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
PARP14 Q460N5 1/20 0.36
KEAP1 Q14145 2/20 0.35
NFE2L2 Q16236 1/20 0.35
SLC6A2 P23975 3/20 0.33
HTR2A P28223 3/20 0.33
HSD17B10 Q99714 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
GLO1 Q04760 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27369292 0.78 GPR84 (0.44) NR3C1NR3C2HTR2AKDM4EALDH1A1
SCHEMBL27965809 0.77 CYP2A6 (0.35) JAK2HTR2A
SCHEMBL27906752 0.77 FFAR1 (0.43) HTR2A
SCHEMBL27524231 0.77 NR4A2 (0.46) NR3C1PGRNR3C2HTR2A
SCHEMBL27771264 0.77 HTR2A (0.44) L3MBTL1HTR2AKDM4EALDH1A1
SCHEMBL28678155 0.76 HTR2A (0.45) HTR2A
SCHEMBL27908791 0.74 HTR2A (0.35) HTR2AKDM4EALDH1A1
SCHEMBL28880740 0.74 PTGS2 (0.43) JAK2
SCHEMBL28818816 0.73 SLC6A4 (0.39) NR3C2HTR2AALDH1A1
SCHEMBL28291599 0.73 POLB (0.37) L3MBTL1SLC6A2HTR2AHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109748840-A A kind of synthetic method of 2- substituted indole derivative 中国医学科学院药物研究所 2019-05-14 CN disclosed