SCHEMBL28332633

SCHEMBL28332633

Nc1cc(F)nc2cccnc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.50
TOP1 P11387 6/20 0.42
HSP90AA1 P07900 4/20 0.40
HSP90AB1 P08238 3/20 0.40
CASP6 P55212 2/20 0.40
KDM4E B2RXH2 2/20 0.39
TP53 P04637 2/20 0.39
MAPT P10636 2/20 0.39
TSHR P16473 2/20 0.39
HTT P42858 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 2/20 0.39
CASP1 P29466 1/20 0.39
ATM Q13315 1/20 0.39
HSD17B10 Q99714 1/20 0.39
LMNA P02545 2/20 0.39
GMNN O75496 1/20 0.39
MMP2 P08253 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23676516 0.81 PRMT5 (0.68) PRMT5TOP1HSP90AA1HSP90AB1CASP6
SCHEMBL30625771 0.78 MMP2 (0.46) PRMT5TOP1HSP90AA1CASP6KDM4E
SCHEMBL6637754 0.78 PRMT5 (0.59) PRMT5TOP1CASP6KDM4EALDH1A1
SCHEMBL9709781 0.74 PRMT5 (0.54) PRMT5TOP1CASP6LMNAHRH4
SCHEMBL2471617 0.73 SLC40A1 (0.47) PRMT5HSP90AA1HSP90AB1CASP6KDM4E
SCHEMBL5822770 0.71 PDE10A (0.45) PRMT5TOP1HSP90AA1HSP90AB1CASP6
SCHEMBL27293402 0.71 NCF1 (0.60) KDM4ETP53MAPTTSHRHTT
SCHEMBL544243 0.70 NCF1 (0.54) PRMT5HSP90AA1HSP90AB1CASP6KDM4E
Hydrochloric Acid SCHEMBL26697692 0.68 NCF1 (0.52) PRMT5HSP90AA1HSP90AB1CASP6KDM4E
SCHEMBL29517215 0.67 DHFR (0.54) PRMT5HSP90AA1KDM4ETP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110386945-A A kind of big ring class kinase inhibitor 成都先导药物开发股份有限公司 2019-10-29 CN disclosed