SCHEMBL28337457

SCHEMBL28337457

COc1cc(OC)cc(-c2cccnc2C=O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.47
ABCB1 P08183 2/20 0.47
BCR P11274 2/20 0.47
CLK4 Q9HAZ1 2/20 0.42
DYRK1A Q13627 1/20 0.42
ERN1 O75460 1/20 0.41
GLO1 Q04760 1/20 0.41
CYP1A1 P04798 3/20 0.41
CYP1B1 Q16678 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2E1 P05181 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C8 P10632 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2A6 P11509 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP4B1 P13584 2/20 0.41
CYP2B6 P20813 2/20 0.41
CYP3A5 P20815 2/20 0.41
CYP2A7 P20853 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7570350 0.88 DYRK1A (0.55) CLK4DYRK1AERN1GLO1CYP1A2
SCHEMBL14484609 0.86 CLK4 (0.51) ABL1ABCB1BCRCLK4CYP2A6
SCHEMBL11617705 0.79 KMT2A (0.46) ERN1TP53TSHRMAPTKMT2A
SCHEMBL27951853 0.79 POLB (0.37) ABL1ERN1CYP1A2CYP2A6CYP2C9
SCHEMBL10119321 0.77 S1PR1 (0.46) CYP3A4TP53MAPT
SCHEMBL2083958 0.76 ERN1 (0.41) ABL1CLK4ERN1NFE2L2
SCHEMBL8512088 0.75 S100A4 (0.45) ABL1ERN1CYP3A4CYP2D6CYP2A6
SCHEMBL2083077 0.74 ALDH1A1 (0.42) ABL1GLO1CYP2A6TSHRMAPT
SCHEMBL2085980 0.74 NFE2L2 (0.46) ERN1CYP1A2CYP3A4CYP2D6TP53
SCHEMBL29889754 0.74 TUBB4A (0.50) ABL1ABCB1BCRCLK4DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110563641-B Ortho-halogenated phenyl pyridine ketone compound and preparation method thereof 三峡大学 2023-03-24 CN disclosed
CN-110563641-A Ortho-halogenated phenyl pyridine ketone compound and preparation method thereof 三峡大学 2019-12-13 CN disclosed