SCHEMBL2838800

SCHEMBL2838800

CCOC(=O)N1CCC(O)c2ccoc2C1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
GPR119 Q8TDV5 1/20 0.41
NOS2 P35228 4/20 0.40
NOS1 P29475 3/20 0.40
GAA P10253 1/20 0.40
NOS3 P29474 1/20 0.40
ALDH1A1 P00352 2/20 0.40
BRD4 O60885 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
POLB P06746 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2835641 0.87 ALDH1A1 (0.38) NPC1L3MBTL1GPR119GAAALDH1A1
SCHEMBL2835764 0.80 GAA (0.40) L3MBTL1NOS2NOS1GAANOS3
SCHEMBL2836018 0.73 OPRK1 (0.33) L3MBTL1
SCHEMBL21767046 0.73 LMNA (0.43) NPC1GAAALDH1A1MEN1KMT2A
SCHEMBL2835727 0.73 L3MBTL1 (0.42) L3MBTL1GAAALDH1A1MEN1KMT2A
SCHEMBL2840999 0.70 KMT2A (0.43) L3MBTL1GAAALDH1A1MEN1KMT2A
SCHEMBL2841889 0.69 OPRM1 (0.35)
SCHEMBL2840528 0.68 CYP3A4 (0.36)
SCHEMBL2837958 0.67 ALDH1A1 (0.36) ALDH1A1MAPT
SCHEMBL1219954 0.65 GAA (0.65) L3MBTL1NOS2GAANOS3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8217031-B2 Heteroaryl derivatives NIPPON SHINYAKU CO., LTD. (JP) 2012-07-10 US disclosed
US-20100048537-A1 HETEROARYL DERIVATIVES NIPPON SHINYAKU CO., LTD. (JP) 2010-02-25 US disclosed
EP-2141168-A1 HETEROARYL DERIVATIVES Nippon Shinyaku Co., Ltd. (JP) 2010-01-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048537-A1 HETEROARYL DERIVATIVES OPRD1, OPRM1, OPRK1 NPC1 1665/4885L3MBTL1 2724/4885GPR119 305/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.