Water

Water

SCHEMBL28396801

O.O=C(O)c1cccc2cccnc12

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 known ✓ P09874 1/20 0.68
CHRM1 known ✓ P11229 1/20 0.52
ADRA1A known ✓ P35348 1/20 0.52
HDAC8 known ✓ Q9BY41 1/20 0.52
MMP8 known ✓ P22894 1/20 0.50
MMP13 known ✓ P45452 1/20 0.50
ALDH1A1 P00352 6/20 0.68
LMNA P02545 3/20 0.68
ALOX12 P18054 2/20 0.68
KDM4E B2RXH2 6/20 0.57
TDP1 Q9NUW8 2/20 0.57
TSHR P16473 4/20 0.55
MAPT P10636 3/20 0.55
CYP3A4 P08684 2/20 0.55
ALOX15 P16050 2/20 0.55
L3MBTL1 Q9Y468 2/20 0.55
BLM P54132 1/20 0.55
AGER Q15109 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
NAPRT Q6XQN6 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29749881 0.98 PARP1 (0.70) PARP1ALDH1A1LMNAALOX12KDM4E
SCHEMBL111826 0.98 PARP1 (0.70) PARP1ALDH1A1LMNAALOX12KDM4E
SCHEMBL16859274 0.96 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12KDM4E
SCHEMBL28875211 0.96 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12KDM4E
Hydrochloric Acid SCHEMBL9691259 0.96 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12KDM4E
SCHEMBL31120780 0.96 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12KDM4E
Hydrochloric Acid SCHEMBL7320778 0.96 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12KDM4E
SCHEMBL30006639 0.96 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12KDM4E
SCHEMBL27534215 0.96 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12KDM4E
SCHEMBL27634251 0.96 PARP1 (0.68) PARP1ALDH1A1LMNAALOX12KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111197182-A Etching solution with silicon oxide corrosion inhibitor and method of use thereof 弗萨姆材料美国有限责任公司 2020-05-26 CN claimed