SCHEMBL28409208

SCHEMBL28409208

CC1=C(C(=O)O)C(C)(c2ccc([N+](=O)[O-])cc2)C(C(=O)O)=C(C)N1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.45
SRD5A2 P31213 1/20 0.41
ACHE P22303 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPK1 P28482 2/20 0.40
CES1 P23141 2/20 0.39
ESPL1 Q14674 1/20 0.39
CES2 O00748 1/20 0.38
RAB9A P51151 1/20 0.38
MAPT P10636 3/20 0.38
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 1/20 0.38
HTR1E P28566 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
S1PR3 Q99500 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9102109 0.83 TP53 (0.47) ACHECES1CES2MAPTALDH1A1
SCHEMBL3394019 0.73 CCR2 (0.43) SRD5A2
SCHEMBL4883866 0.71 TP53 (0.43) TDP1ACHECES1CES2MAPT
SCHEMBL3392997 0.71 TDP1 (0.40) TDP1SRD5A2ACHEHSD17B10MAPK1
SCHEMBL4756165 0.70 TP53 (0.43) TDP1ACHEMAPK1CES1CES2
Acetic Acid SCHEMBL27877969 0.67 MAPK1 (0.71) TDP1SRD5A2ACHEHSD17B10MAPK1
Hydrogen Peroxide SCHEMBL28789390 0.66 ALDH1A1 (0.72) TDP1SRD5A2ACHEHSD17B10MAPK1
4-Nitrotoluene SCHEMBL30483931 0.66 ACHE (0.82) TDP1SRD5A2ACHEHSD17B10MAPK1
4-Nitrotoluene SCHEMBL9037550 0.66 ACHE (0.82) TDP1SRD5A2ACHEHSD17B10MAPK1
SCHEMBL4758043 0.66 CRHBP (0.40) TDP1MAPK1MAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111110854-A Composition comprising a histamine release-promoting substance and an inhibitory compound 黄泳华 2020-05-08 CN claimed
CN-111110854-A Composition comprising a histamine release-promoting substance and an inhibitory compound 黄泳华 2020-05-08 CN disclosed