SCHEMBL28443183

SCHEMBL28443183

COC(=O)c1ccc2c(nnn2C)c1CBr

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.35
ALDH1A1 P00352 3/20 0.35
NR4A2 P43354 3/20 0.35
HCAR3 P49019 1/20 0.35
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
LMNA P02545 2/20 0.34
TP53 P04637 2/20 0.34
MAPT P10636 4/20 0.34
HSD17B10 Q99714 2/20 0.34
HPGD P15428 2/20 0.34
HTT P42858 1/20 0.34
POLB P06746 1/20 0.33
AHR P35869 1/20 0.33
CCKBR P32239 1/20 0.33
PTGER4 P35408 1/20 0.33
GLA P06280 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8953225 0.80 KDM4E (0.38) KDM4EALDH1A1NR4A2HCAR3NPC1
SCHEMBL28897492 0.79 L3MBTL1 (0.41) KDM4EALDH1A1NR4A2NPC1RAB9A
SCHEMBL2013415 0.76 NR4A2 (0.45) KDM4EALDH1A1NR4A2NPC1RAB9A
SCHEMBL17910027 0.70 KMT2A (0.37) KDM4EALDH1A1NR4A2HCAR3HSD17B10
SCHEMBL30618046 0.70 KMT2A (0.37) KDM4EALDH1A1NR4A2HCAR3HSD17B10
SCHEMBL28448806 0.69 KMT2A (0.41) KDM4EALDH1A1NPC1RAB9ALMNA
SCHEMBL28448807 0.69 ALDH1A1 (0.41) KDM4EALDH1A1RAB9ASMN1; SMN2LMNA
SCHEMBL29041518 0.69 LMNA (0.52) KDM4EALDH1A1LMNAMAPTHSD17B10
SCHEMBL1354809 0.69 KDM4E (0.38) KDM4EALDH1A1NR4A2NPC1RAB9A
SCHEMBL8524627 0.68 NNMT (0.39) KDM4EALDH1A1HCAR3NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111606928-A Azacyclodiketone compound and preparation method thereof 维清生物科技(上海)有限公司 2020-09-01 CN disclosed