SCHEMBL28459748

SCHEMBL28459748

COC(=O)C(NC(=O)C1(O)C=CC(c2ccccc2)=CC1)C(C)(C)NC(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 2/20 0.36
CTSS P25774 3/20 0.36
CTSK P43235 2/20 0.36
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
PPARA Q07869 5/20 0.33
PPARG P37231 4/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
ITGA4 P13612 1/20 0.32
ITGB7 P26010 1/20 0.32
ACE P12821 1/20 0.32
ATM Q13315 1/20 0.32
AKT1 P31749 1/20 0.32
PPARD Q03181 2/20 0.32
PSEN1 P49768 2/20 0.32
PSEN2 P49810 2/20 0.32
APH1B Q8WW43 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28461037 0.93 CTSS (0.36) CTSSCTSKCTSLCTSBPPARA
SCHEMBL5983441 0.72 NFKB1 (0.36) CTSSCTSKCTSLCTSBNFKB1
SCHEMBL8970782 0.71 MEN1 (0.38) TSHR
Methane SCHEMBL27537449 0.69 NFKB1 (0.36) CTSSCTSKCTSLCTSBNFKB1
SCHEMBL13244981 0.69 SYK (0.58) KLK5CTSSCTSKCTSLCTSB
SCHEMBL13337480 0.69 SYK (0.58) KLK5CTSSCTSKCTSLCTSB
SCHEMBL23787015 0.69 BCL2 (0.36) KLK5PPARAPPARGTSHRATM
SCHEMBL5983320 0.68 ALDH1A1 (0.34) KLK5CTSSCTSKCTSLCTSB
SCHEMBL1119645 0.67 THRB (0.35)
SCHEMBL24234472 0.67 SYK (0.49) KLK5CTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105777464-B Hydroxamic acid derivative and preparation method and application thereof 中国科学院上海药物研究所 2020-09-29 CN disclosed