SCHEMBL28503586

SCHEMBL28503586

O=C(NCCC1CNCCO1)c1ccc2nc(-c3ccccc3)n(Cc3ccccc3)c2c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 8/20 0.51
ACSS2 Q9NR19 6/20 0.44
PDE2A O00408 1/20 0.42
PDE6D O43924 1/20 0.42
ALDH1A1 P00352 1/20 0.42
ALDH2 P05091 1/20 0.42
ALDH3A1 P30838 1/20 0.42
HRH3 Q9Y5N1 1/20 0.41
DRD2 P14416 1/20 0.41
TBXA2R P21731 1/20 0.41
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28503588 0.82 BRD4 (0.42) BRD4ACSS2PDE6DALDH1A1ALDH2
SCHEMBL28503584 0.79 PIK3CA (0.62) PDE2AALDH1A1
SCHEMBL28507636 0.77 ACSS2 (0.59) BRD4ACSS2PDE2APDE6DALDH1A1
SCHEMBL28514126 0.76 PDE6D (0.47) BRD4ACSS2PDE2APDE6DALDH1A1
SCHEMBL28513264 0.75 TP53 (0.53) BRD4PDE2APDE6DALDH1A1ALDH2
SCHEMBL28516171 0.75 THRB (0.50) BRD4PDE2APDE6DALDH1A1ALDH2
SCHEMBL28001720 0.75 BRD4 (0.54) BRD4
SCHEMBL28503579 0.74 ALDH1A1 (0.63) BRD4ACSS2PDE6DALDH1A1ALDH2
SCHEMBL28510581 0.74 SMN1; SMN2 (0.59) ACSS2PDE2A
SCHEMBL28505411 0.73 DRD2 (0.66) BRD4ACSS2PDE6DALDH1A1ALDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107311933-B Benzimidazole derivative, preparation method and application thereof 中国人民解放军军事医学科学院毒物药物研究所 2020-12-22 CN disclosed