SCHEMBL28509099

SCHEMBL28509099

Clc1cc(Cl)c2c[c]ccc2n1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
HIF1A Q16665 1/20 0.35
LMNA P02545 1/20 0.34
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
USP2 O75604 1/20 0.31
HTT P42858 1/20 0.31
ESRRB O95718 1/20 0.31
ESR1 P03372 1/20 0.31
ESRRA P11474 1/20 0.31
ESR2 Q92731 1/20 0.31
NT5E P21589 1/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20476372 0.85 KDM4E (0.32) KDM4ECYP3A4CYP2C19HIF1ALMNA
SCHEMBL6986503 0.81 ESR1 (0.36) LMNAMAOAMAOBESRRBESR1
SCHEMBL693400 0.79 NT5E (0.55) KDM4ENT5EMAPT
SCHEMBL397020 0.71 MAOA (0.54) KDM4ECYP3A4CYP2C19MAOAMAOB
SCHEMBL29420516 0.71 MAOA (0.54) KDM4ECYP3A4CYP2C19MAOAMAOB
SCHEMBL6995818 0.71 ALDH1A1 (0.40) KDM4ELMNAMAPT
SCHEMBL4455983 0.71 AXL (0.37) KDM4ECYP2C19MAPT
SCHEMBL15516443 0.70 KDM4E (0.47) KDM4ECYP3A4CYP2C19HIF1ALMNA
SCHEMBL865202 0.69 CRHBP (0.32)
SCHEMBL29799170 0.69 LMNA (0.46) KDM4ECYP3A4CYP2C19HIF1ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112204010-B Heterocyclic derivatives and uses thereof C&C新药研究所 2024-03-19 CN disclosed
CN-112204010-A Heterocyclic derivatives and use thereof C&C新药研究所 2021-01-08 CN disclosed