SCHEMBL2853364

SCHEMBL2853364

O=C(NCc1cccc(-c2ccccc2)c1)Oc1cnn(-c2ccc([N+](=O)[O-])cc2)c1C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 5/20 0.52
KEAP1 Q14145 1/20 0.45
NFE2L2 Q16236 1/20 0.45
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ATG4B Q9Y4P1 1/20 0.41
EPHX1 P07099 2/20 0.41
FFAR1 O14842 1/20 0.40
ACHE P22303 3/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ACKR3 P25106 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2861197 0.92 CCR1 (0.51) CCR1NPC1MAPTRAB9ANPSR1
SCHEMBL2856304 0.90 KEAP1 (0.53) CCR1KEAP1NFE2L2MAPTEPHX1
SCHEMBL2856460 0.90 CCR1 (0.65) CCR1NPC1MAPTRAB9ANPSR1
SCHEMBL2854462 0.89 KEAP1 (0.48) CCR1KEAP1NFE2L2MAPTEPHX1
SCHEMBL2856294 0.88 CCR1 (0.49) CCR1KEAP1NFE2L2EPHX1KDM4E
SCHEMBL2859089 0.86 ATG4B (0.43) CCR1KEAP1NFE2L2ATG4BEPHX1
SCHEMBL2860700 0.86 KEAP1 (0.46) CCR1KEAP1NFE2L2EPHX1KDM4E
SCHEMBL2856514 0.85 CCR1 (0.49) CCR1NPC1MAPTRAB9ANPSR1
SCHEMBL2858076 0.85 MAPT (0.56) CCR1NPC1MAPTRAB9ANPSR1
SCHEMBL2850321 0.85 SMN1; SMN2 (0.47) CCR1NPC1MAPTRAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed