SCHEMBL2856294

SCHEMBL2856294

O=C(NCc1cccc(-c2ccccc2)c1)Oc1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 9/20 0.49
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
EPHX1 P07099 2/20 0.43
ABCB1 P08183 2/20 0.43
LIPG Q9Y5X9 1/20 0.43
ADAMTS5 Q9UNA0 1/20 0.42
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2856304 0.93 KEAP1 (0.53) CCR1KEAP1NFE2L2EPHX1KDM4E
SCHEMBL2854462 0.92 KEAP1 (0.48) CCR1KEAP1NFE2L2EPHX1KDM4E
SCHEMBL2853388 0.92 CCR1 (0.48) CCR1ABCB1KDM4EALDH1A1
SCHEMBL2860700 0.89 KEAP1 (0.46) CCR1KEAP1NFE2L2EPHX1KDM4E
SCHEMBL2849956 0.89 CCR1 (0.62) CCR1
SCHEMBL2853253 0.89 KEAP1 (0.42) CCR1KEAP1NFE2L2EPHX1LIPG
SCHEMBL2854543 0.88 CCR1 (0.54) CCR1ABCB1
SCHEMBL2853364 0.88 CCR1 (0.52) CCR1KEAP1NFE2L2EPHX1KDM4E
SCHEMBL2856356 0.88 ALDH1A1 (0.47) CCR1ABCB1KDM4EALDH1A1
SCHEMBL2859076 0.86 KEAP1 (0.42) CCR1KEAP1NFE2L2EPHX1LIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed