SCHEMBL2860700

SCHEMBL2860700

COc1ccc(-n2ncc(OC(=O)NCc3cccc(-c4ccccc4)c3)c2C(F)(F)F)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
DGAT2 Q96PD7 2/20 0.45
EPHX1 P07099 2/20 0.44
USP2 O75604 1/20 0.41
POLB P06746 1/20 0.41
TP53 P04637 1/20 0.41
CCR1 P32246 3/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SMO Q99835 1/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
LMNA P02545 1/20 0.40
DHODH Q02127 2/20 0.40
SENP1 Q9P0U3 1/20 0.40
CHRM3 P20309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2856304 0.92 KEAP1 (0.53) KEAP1NFE2L2DGAT2EPHX1POLB
SCHEMBL2852520 0.92 TP53 (0.47) DGAT2POLBTP53KDM4EALDH1A1
SCHEMBL2854462 0.90 KEAP1 (0.48) KEAP1NFE2L2EPHX1CCR1KDM4E
SCHEMBL2854330 0.89 CCR1 (0.52) USP2POLBCCR1
SCHEMBL2856294 0.89 CCR1 (0.49) KEAP1NFE2L2EPHX1CCR1KDM4E
SCHEMBL2853364 0.86 CCR1 (0.52) KEAP1NFE2L2EPHX1CCR1KDM4E
SCHEMBL2853277 0.86 CCR1 (0.50) DGAT2POLBTP53CCR1SMN1; SMN2
SCHEMBL2852633 0.84 TAAR1 (0.57) TP53KDM4EALDH1A1LMNA
SCHEMBL2852545 0.84 NPBWR1 (0.42) USP2POLBTP53CCR1KDM4E
SCHEMBL2856625 0.84 TSHR (0.48) CCR1SMN1; SMN2SMOLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed