SCHEMBL2854496

SCHEMBL2854496

O=C(NCCc1c(Cl)cccc1Cl)Oc1cnn(-c2ccc(F)cc2)c1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.47
TRPV1 Q8NER1 1/20 0.40
CCR1 P32246 3/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPT P10636 1/20 0.38
NR3C1 P04150 5/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
TRPC3 Q13507 1/20 0.37
NPSR1 Q6W5P4 2/20 0.37
DGAT2 Q96PD7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2858618 0.93 ALDH1A1 (0.41) P2RX7TRPV1CCR1ALDH1A1KDM4E
SCHEMBL2854705 0.92 ALDH1A1 (0.46) P2RX7TRPV1ALDH1A1KDM4EMAPT
SCHEMBL2848315 0.90 TRPV1 (0.54) P2RX7TRPV1ALDH1A1KDM4EMAPT
SCHEMBL2853063 0.90 P2RX7 (0.48) P2RX7TRPV1CCR1ALDH1A1KDM4E
SCHEMBL2857996 0.86 CCR1 (0.48) P2RX7TRPV1CCR1ALDH1A1KDM4E
SCHEMBL2863154 0.86 MAPT (0.45) P2RX7CCR1ALDH1A1KDM4EMAPT
SCHEMBL2853186 0.85 TRPV1 (0.41) P2RX7TRPV1KDM4EMAPTNPSR1
SCHEMBL2860458 0.85 TP53 (0.46) P2RX7MAPTNR3C1NPSR1
SCHEMBL2850857 0.85 TP53 (0.46) P2RX7MAPTNR3C1NPSR1
SCHEMBL2854346 0.85 MAPT (0.52) P2RX7CCR1ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed