SCHEMBL2860106

SCHEMBL2860106

O=C(NCc1ccccc1)Oc1cnn(Cc2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 2/20 0.52
EPHX1 P07099 2/20 0.46
MGLL Q99685 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HDAC3 O15379 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
NCOR2 Q9Y618 1/20 0.44
SCD O00767 4/20 0.44
SCD5 Q86SK9 3/20 0.44
ALDH1A1 P00352 2/20 0.44
ITK Q08881 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM5C P41229 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2852927 0.94 KLKB1 (0.50) KLKB1NPC1RAB9AL3MBTL1ALDH1A1
SCHEMBL2848515 0.93 LMNA (0.50) KLKB1NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL2861622 0.91 EPHX1 (0.60) EPHX1L3MBTL1SMN1; SMN2
SCHEMBL2853080 0.88 LMNA (0.50) KLKB1NPC1RAB9AL3MBTL1SCD5
SCHEMBL2852519 0.87 TAAR1 (0.59) KLKB1NPC1RAB9AL3MBTL1HDAC3
SCHEMBL2859721 0.87 KLKB1 (0.49) KLKB1RAB9AL3MBTL1SCDSCD5
SCHEMBL2860989 0.84 ALDH1A1 (0.68) NPC1RAB9ASCD5ALDH1A1SMN1; SMN2
SCHEMBL2859353 0.82 TAAR1 (0.66) NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL18544527 0.81 KLKB1 (0.68) KLKB1
SCHEMBL2852630 0.81 TAAR1 (0.52) NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed