SCHEMBL2860652

SCHEMBL2860652

COc1ccc(-n2ncc(OC(=O)NCCc3ccc(C)cc3C)c2C)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.44
TDP1 Q9NUW8 3/20 0.44
BLM P54132 1/20 0.44
NR2F2 P24468 2/20 0.42
NPC1 O15118 5/20 0.42
RAB9A P51151 4/20 0.42
THRB P10828 1/20 0.42
GALR3 O60755 1/20 0.42
MAPT P10636 4/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
NPBWR1 P48145 1/20 0.40
MCHR1 Q99705 1/20 0.40
TP53 P04637 2/20 0.40
GAA P10253 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
PKM P14618 1/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2857276 0.89 RAB9A (0.47) NPC1RAB9ATHRBMAPTSMN1; SMN2
SCHEMBL2850323 0.88 MAPT (0.47) POLBTDP1NPC1RAB9AMAPT
SCHEMBL2857343 0.85 P2RX7 (0.42) THRBMAPTSMN1; SMN2NPBWR1TP53
SCHEMBL2858680 0.83 NPC1 (0.45) NPC1RAB9AMAPTSMN1; SMN2NFKB1
SCHEMBL2853389 0.82 NPC1 (0.62) NPC1RAB9ATHRBMAPTSMN1; SMN2
SCHEMBL2861643 0.80 CNR1 (0.50) POLBNPC1RAB9ASMN1; SMN2TP53
SCHEMBL2861634 0.79 RAB9A (0.44) NPC1RAB9AMAPTSMN1; SMN2NFKB1
SCHEMBL2857875 0.79 P2RX7 (0.45) MAPTSMN1; SMN2TP53
SCHEMBL2854836 0.79 MAPK14 (0.42) NPC1RAB9AMAPTGAAPKM
SCHEMBL2858128 0.78 ALDH1A1 (0.46) POLBNPC1RAB9AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed