SCHEMBL2861180

SCHEMBL2861180

Cc1cccc(CNC(=O)[CH]COC(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.46
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
OPRM1 P35372 1/20 0.42
CYP2D6 P10635 1/20 0.42
FBP1 P09467 1/20 0.41
TP53 P04637 1/20 0.41
ASAH1 Q13510 2/20 0.40
ADORA2A P29274 2/20 0.40
ROCK2 O75116 1/20 0.40
ADORA1 P30542 1/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2856255 0.85 GAA (0.48) ALDH1A1
SCHEMBL2858150 0.84 LMNA (0.52) ALDH1A1KDM4EHPGDTP53KMT2A
SCHEMBL2851648 0.84 ALDH1A1 (0.51) ALDH1A1HPGDCYP2D6MMP1MMP2
SCHEMBL2857248 0.79 CARM1 (0.39) ALDH1A1ROCK2
SCHEMBL2861183 0.78 TP53 (0.47) MMP13ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL2854435 0.77 TSHR (0.48) ALDH1A1HPGDTP53KMT2A
SCHEMBL6581126 0.75 MMP13 (0.55) MMP13ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL4971087 0.74 MMP13 (0.43) MMP13ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL2858022 0.74 CA12 (0.49) MMP13ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL4971081 0.74 MMP13 (0.43) MMP13ALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963277-B1 FLUORINATED COMPOUNDS NPS PHARMA INC (US) 2010-01-20 EP claimed
EP-1963277-B1 FLUORINATED COMPOUNDS NPS PHARMA INC (US) 2010-01-20 EP disclosed