SCHEMBL2851648

SCHEMBL2851648

O=C([CH]COC(F)F)NCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
LMNA P02545 4/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
MMP1 P03956 3/20 0.49
MMP2 P08253 3/20 0.49
MMP9 P14780 3/20 0.49
CYP2C9 P11712 1/20 0.48
MAPT P10636 3/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TSHR P16473 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ATM Q13315 1/20 0.43
GAA P10253 1/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854435 0.87 TSHR (0.48) ALDH1A1LMNAMAPTL3MBTL1HTT
SCHEMBL2858150 0.85 LMNA (0.52) ALDH1A1LMNAMAPTL3MBTL1SMN1; SMN2
SCHEMBL2861180 0.84 MMP13 (0.46) ALDH1A1CYP2D6MMP1MMP2MMP9
SCHEMBL2856255 0.84 GAA (0.48) ALDH1A1L3MBTL1HTTNPSR1GAA
SCHEMBL2852748 0.80 GRM5 (0.40) LMNAHPGD
SCHEMBL2849991 0.77 RECQL (0.51) ALDH1A1LMNAMAPTHTTTSHR
SCHEMBL4073041 0.75 ALDH1A1 (0.62) ALDH1A1LMNACYP2D6CYP2C19MMP1
SCHEMBL27839057 0.75 ALDH1A1 (0.62) ALDH1A1LMNACYP2D6CYP2C19MMP1
SCHEMBL2851650 0.74 TSHR (0.63) ALDH1A1LMNACYP2C19L3MBTL1HTT
SCHEMBL1416058 0.74 ALDH1A1 (0.61) ALDH1A1LMNACYP2D6CYP2C19MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963277-B1 FLUORINATED COMPOUNDS NPS PHARMA INC (US) 2010-01-20 EP claimed
US-7902401-B2 Fluorinated compounds NPS PHARMACEUTICALS, INC. (US) 2011-03-08 US disclosed
EP-1963277-B1 FLUORINATED COMPOUNDS NPS PHARMA INC (US) 2010-01-20 EP disclosed