SCHEMBL2862091

SCHEMBL2862091

CCCc1c(C(=O)NCc2ccc(OC)cc2OC)cnn1-c1ccc(Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
MAPT P10636 4/20 0.53
MAPK1 P28482 1/20 0.49
TAS1R3 Q7RTX0 2/20 0.49
TAS1R1 Q7RTX1 2/20 0.49
MAPK14 Q16539 1/20 0.47
TSHR P16473 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
GAA P10253 2/20 0.47
PKM P14618 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
CCR1 P32246 1/20 0.45
KLKB1 P03952 1/20 0.45
LMNA P02545 1/20 0.45
TP53 P04637 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850782 0.86 ALDH1A1 (0.42) ALDH1A1MAPTTAS1R3TAS1R1TSHR
SCHEMBL2850622 0.83 ALDH1A1 (0.57) ALDH1A1MAPTMAPK1MAPK14GAA
SCHEMBL2856684 0.77 TAS1R3 (0.58) ALDH1A1MAPTTAS1R3TAS1R1TSHR
SCHEMBL4670752 0.77 CCR1 (0.49) ALDH1A1MAPTMAPK1MAPK14GAA
SCHEMBL4672609 0.77 CCR1 (0.50) ALDH1A1MAPTMAPK1MAPK14GAA
SCHEMBL2850896 0.75 DGAT2 (0.57) ALDH1A1MAPTTAS1R3TAS1R1TSHR
SCHEMBL2857376 0.75 ALDH1A1 (0.67) ALDH1A1MAPTMAPK1MAPK14GAA
SCHEMBL2856352 0.74 DGAT2 (0.56) ALDH1A1MAPTTAS1R3TAS1R1TSHR
SCHEMBL2853245 0.74 ALDH1A1 (0.68) ALDH1A1MAPTMAPK1MAPK14GAA
SCHEMBL2854156 0.73 ROCK2 (0.46) ALDH1A1MAPTTSHRNPSR1KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed