SCHEMBL28626906

SCHEMBL28626906

CCC(=O)Oc1c(C)n(C)c2ccc(C(F)(F)F)cc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.45
AKR1B1 P15121 1/20 0.44
KDM4E B2RXH2 1/20 0.41
ALOX5 P09917 1/20 0.40
SRC P12931 1/20 0.40
KIF11 P52732 1/20 0.39
RORA P35398 1/20 0.38
RORC P51449 1/20 0.38
RORB Q92753 1/20 0.38
POLB P06746 2/20 0.37
HTT P42858 1/20 0.37
AKR1C3 P42330 1/20 0.37
CYP2C9 P11712 1/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
PDE4A P27815 3/20 0.36
PDE4B Q07343 3/20 0.36
PDE4C Q08493 3/20 0.36
PDE4D Q08499 3/20 0.36
PTGER4 P35408 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30675225 1.00 PTGDR2 (0.45) PTGDR2AKR1B1KDM4EALOX5SRC
SCHEMBL28628728 0.83 LMNA (0.43) KDM4EPOLBHTTCYP2C9
SCHEMBL29123399 0.75 POLB (0.37) KDM4EALOX5RORCPOLB
SCHEMBL30792537 0.74 LMNA (0.42) KDM4ERORARORCRORBPOLB
SCHEMBL28626909 0.73 AKR1C3 (0.47) PTGDR2AKR1B1KDM4EALOX5SRC
SCHEMBL18015724 0.73 KIF11 (0.50) PTGDR2AKR1B1KDM4EALOX5SRC
SCHEMBL16729412 0.72 KIF11 (0.51) PTGDR2KDM4ESRCKIF11CYP2C9
SCHEMBL17968711 0.72 KIF11 (0.49) PTGDR2KDM4ESRCKIF11RORA
SCHEMBL28637173 0.71 AKR1C3 (0.45) PTGDR2SRCKIF11AKR1C3CYP2C9
SCHEMBL4616695 0.71 ALOX5 (0.50) KDM4EALOX5SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429332-B 3-substituted indole derivative, preparation method thereof and application thereof in antitumor drugs 长春工业大学 2023-12-15 CN disclosed
CN-113429332-A 3-substituted indole derivative, preparation method thereof and application thereof in antitumor drugs 长春工业大学 2021-09-24 CN disclosed