SCHEMBL2863699

SCHEMBL2863699

CCc1cc(Br)ccc1O[Si](C)(C)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HTT P42858 1/20 0.40
GAA P10253 1/20 0.39
NPY1R P25929 1/20 0.39
NPY2R P49146 1/20 0.39
DRD2 P14416 1/20 0.38
TSHR P16473 3/20 0.38
PTGDR2 Q9Y5Y4 2/20 0.38
GLA P06280 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
APLNR P35414 2/20 0.36
HPGD P15428 1/20 0.36
POLB P06746 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9585824 0.84 GAA (0.40) MEN1KMT2AHTTGAANPY1R
SCHEMBL15514887 0.82 DRD2 (0.38) MEN1KMT2AHTTGAADRD2
SCHEMBL2401781 0.81 DRD2 (0.43) MEN1KMT2AHTTGAADRD2
SCHEMBL6519564 0.78 ALDH1A1 (0.44) MEN1KMT2AHTTGAADRD2
SCHEMBL4471859 0.78 EDNRB (0.36) MEN1KMT2AHTTGAANPY1R
SCHEMBL6448162 0.78 PTGDR2 (0.39) MEN1KMT2AHTTGAANPY1R
SCHEMBL30393256 0.77 RAB9A (0.43) MEN1KMT2ADRD2TSHRPTGDR2
SCHEMBL2287094 0.77 RAB9A (0.43) MEN1KMT2ADRD2TSHRPTGDR2
SCHEMBL9853837 0.77 L3MBTL1 (0.44) KMT2ADRD2HPGDKDM4E
SCHEMBL2850545 0.77 MEN1 (0.42) MEN1KMT2AHTTDRD2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1456160-B1 VITAMIN D ANALOGUES GALDERMA RES & DEV (FR) 2010-01-20 EP disclosed
US-6924400-B2 Triaromatic vitamin D analogues GALDERMA RESEARCH & DEVELOPMENT, SNC (FR) 2005-08-02 US disclosed
EP-1456160-A2 VITAMIN D ANALOGUES Galderma Research & Development, S.N.C. (FR) 2004-09-15 EP disclosed
US-20030195259-A1 Triaromatic vitamin D analogues GALDERMA RESEARCH & DEVELOPMENT (FR) 2003-10-16 US disclosed
WO-2003050067-A2 VITAMIN D ANALOGUES GALDERMA RESEARCH & DEVELOPMENT, SNC (FR) 2003-06-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030195259-A1 Triaromatic vitamin D analogues CYP24A1, CYP2R1, VDR MEN1 945/4885KMT2A 4353/4885HTT 2386/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.