SCHEMBL287259

SCHEMBL287259

COc1ccc(C(=O)CN(NS(=O)(=O)c2ccc(C)cc2)C(=O)C2CCCNC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
ALDH1A1 P00352 4/20 0.40
MAPT P10636 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
EGFR P00533 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL286982 0.89 KMT2A (0.41) KMT2AMEN1ALDH1A1MAPTCYP1A2
SCHEMBL287097 0.87 MMP1 (0.38) ALDH1A1MAPTMMP1MMP9MMP13
SCHEMBL287365 0.72 NPY5R (0.41) KMT2AALDH1A1MAPTCYP1A2HPGD
SCHEMBL287774 0.71 USP30 (0.36) ALDH1A1MAPTHPGDHTT
SCHEMBL6563603 0.70 KEAP1 (0.45) KMT2AALDH1A1MAPTHPGDLMNA
SCHEMBL11798075 0.69 NPC1 (0.59) KMT2AMEN1ALDH1A1LMNANPC1
SCHEMBL284518 0.68 ALDH1A1 (0.34) KMT2AMEN1ALDH1A1MAPTLMNA
SCHEMBL7943813 0.67 ALDH1A1 (0.57) KMT2AMEN1ALDH1A1MAPTHPGD
SCHEMBL287828 0.66 ALDH1A1 (0.38) KMT2AMEN1ALDH1A1CYP1A2HPGD
SCHEMBL287258 0.65 ALDH1A1 (0.52) KMT2AMEN1ALDH1A1NPC1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427432-A2 NOVEL HETEROCYCLIC COMPOUNDS Torrent Pharmaceuticals Limited (IN) 2012-03-14 EP claimed
WO-2010128528-A2 NOVEL HETEROCYCLIC COMPOUNDS TORRENT PHARMACEUTICALS LIMITED (IN) 2010-11-11 WO claimed
EP-2427432-A2 NOVEL HETEROCYCLIC COMPOUNDS Torrent Pharmaceuticals Limited (IN) 2012-03-14 EP disclosed
WO-2010128528-A2 NOVEL HETEROCYCLIC COMPOUNDS TORRENT PHARMACEUTICALS LIMITED (IN) 2010-11-11 WO disclosed