SCHEMBL286982

SCHEMBL286982

Cc1ccc(S(=O)(=O)NN(CC(=O)c2ccccc2)C(=O)C2CCCNC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
REN P00797 4/20 0.41
TSHR P16473 1/20 0.40
RECQL P46063 1/20 0.40
ALDH1A1 P00352 4/20 0.38
MEN1 O00255 2/20 0.38
CYP2C9 P11712 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MAPT P10636 1/20 0.36
CA12 O43570 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
ATM Q13315 1/20 0.36
CA9 Q16790 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL287259 0.89 KMT2A (0.40) KMT2ATSHRALDH1A1MEN1CYP2C9
SCHEMBL287365 0.80 NPY5R (0.41) KMT2ATSHRALDH1A1MAPTCYP1A2
SCHEMBL287774 0.76 USP30 (0.36) ALDH1A1NPSR1MAPT
SCHEMBL287097 0.74 MMP1 (0.38) RENALDH1A1MAPTPOLB
SCHEMBL284518 0.71 ALDH1A1 (0.34) KMT2ARENTSHRRECQLALDH1A1
SCHEMBL287828 0.71 ALDH1A1 (0.38) KMT2ARENTSHRALDH1A1MEN1
SCHEMBL287108 0.69 RAB9A (0.39) KMT2ATSHRALDH1A1MEN1NPC1
SCHEMBL286983 0.68 ALDH1A1 (0.40) KMT2ARENTSHRALDH1A1MEN1
SCHEMBL25269242 0.67 SLC6A1 (0.46) KMT2ATSHRALDH1A1MAPTATM
SCHEMBL7001156 0.65 KMT2A (0.64) KMT2ATSHRMEN1MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427432-A2 NOVEL HETEROCYCLIC COMPOUNDS Torrent Pharmaceuticals Limited (IN) 2012-03-14 EP claimed
WO-2010128528-A2 NOVEL HETEROCYCLIC COMPOUNDS TORRENT PHARMACEUTICALS LIMITED (IN) 2010-11-11 WO claimed
EP-2427432-A2 NOVEL HETEROCYCLIC COMPOUNDS Torrent Pharmaceuticals Limited (IN) 2012-03-14 EP disclosed
WO-2010128528-A2 NOVEL HETEROCYCLIC COMPOUNDS TORRENT PHARMACEUTICALS LIMITED (IN) 2010-11-11 WO disclosed