SCHEMBL28750554

SCHEMBL28750554

COC(=O)C(NC(=N)N)C1CCc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.43
USP2 O75604 1/20 0.41
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
PIN1 Q13526 1/20 0.39
ADORA2A P29274 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
IDO1 P14902 1/20 0.36
PDPK1 O15530 1/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ECE1 P42892 5/20 0.36
SLC5A7 Q9GZV3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27583416 0.89 ALDH1A1 (0.39) TSHRUSP2KMT2AMEN1ALDH1A1
SCHEMBL27649366 0.86 ECE1 (0.41) ALDH1A1ECE1
SCHEMBL23699443 0.75 USP2 (0.43) TSHRUSP2PDE4APDE4BPDE4C
SCHEMBL12924867 0.75 SLC6A3 (0.51) TSHRKMT2AALDH1A1
SCHEMBL23699381 0.74 TSHR (0.44) TSHRUSP2PDE4APDE4BPDE4C
SCHEMBL23934503 0.72 USP2 (0.45) TSHRUSP2PDE4APDE4BPDE4C
SCHEMBL17335654 0.71 TRPM8 (0.44) PIN1IDO1PDPK1
SCHEMBL15882481 0.71 TRPM8 (0.44) PIN1IDO1PDPK1
SCHEMBL31757665 0.71 DRD2 (0.41) IDO1MAPTALDH1A1
SCHEMBL31758027 0.71 DRD2 (0.41) IDO1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1396906-A Calcilytic compounds SMITHKLINE BEECHAM CORP (US) 2003-02-12 CN disclosed