SCHEMBL28787308

SCHEMBL28787308

Cc1ccc(C2CCN(OC(=O)C(C)(C)C)CC2)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 2/20 0.42
GPR119 Q8TDV5 3/20 0.41
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
PDK2 Q15119 7/20 0.36
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
OPRL1 P41146 1/20 0.35
PRCP P42785 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
SLC9A1 P19634 1/20 0.34
CYP2C19 P33261 1/20 0.34
KCNH2 Q12809 1/20 0.34
APLNR P35414 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28024911 0.86 GPR119 (0.40) DRD4GPR119OPRL1SLC6A3CYP3A4
SCHEMBL27790080 0.83 RBP4 (0.46) GPR119MAPTOPRL1SLC6A2SLC6A4
SCHEMBL28146205 0.79 RBP4 (0.48) OPRL1SLC6A3CYP3A4CYP2C9SLC9A1
SCHEMBL28146200 0.78 RBP4 (0.50)
SCHEMBL28146207 0.78 RBP4 (0.48) CYP3A4CYP2C9CYP2C19
SCHEMBL28024448 0.77 OPRL1 (0.36) DRD4LMNAMAPTTHRBOPRL1
SCHEMBL28147246 0.76 RBP4 (0.49) CYP3A4CYP2C9SLC9A1CYP2C19KCNH2
SCHEMBL27704480 0.75 DRD2 (0.46) GPR119DRD2KCNH2
SCHEMBL28766839 0.74 MAPT (0.40) DRD4DRD2DRD3MAPTPTGDR2
SCHEMBL14924438 0.74 OPRL1 (0.46) DRD4OPRL1SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101778831-A Novel piperazine amide derivatives HOFFMANN LA ROCHE 2010-07-14 CN disclosed