SCHEMBL28794072

SCHEMBL28794072

N#Cc1cc(-c2ccc(F)cc2)[nH]c1C[SH](=O)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
GCGR P47871 3/20 0.38
MAPK14 Q16539 3/20 0.38
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
CTSV O60911 1/20 0.35
CTSL P07711 1/20 0.35
PTK2 Q05397 2/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
CCNB2 O95067 1/20 0.34
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL194128 0.70 AXL (0.45) MAPTKMT2AKDM4EALDH1A1GAA
SCHEMBL194942 0.70 PTGS2 (0.47) MAPTKMT2AKDM4EALDH1A1GAA
SCHEMBL27575026 0.67 MAOA (0.41) MAOAMAOBCYP11B1CYP11B2
SCHEMBL28220967 0.67 ERCC1 (0.46) MAPTKMT2AALDH1A1GAACTSV
SCHEMBL11737297 0.66 ERCC1 (0.57) MAPTKMT2AKDM4EALDH1A1GAA
SCHEMBL1463119 0.62 CYP11B2 (0.49) KMT2AKDM4EALDH1A1GCGRMAPK14
SCHEMBL15018349 0.61 TRPV4 (0.52) MAOAMAOBCYP11B1CYP11B2
SCHEMBL17827370 0.60 CYP11B2 (0.59) KMT2AKDM4EALDH1A1HTTMAOA
SCHEMBL194510 0.60 ALDH1A1 (0.51) MAPTKMT2AKDM4EALDH1A1GAA
SCHEMBL194615 0.60 ALDH1A1 (0.48) MAPTKMT2AKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105524046-A Process for producing pyrrole compound TAKEDA PHARMACEUTICAL 2016-04-27 CN disclosed
CN-102421753-B Process for preparing azole compounds TAKEDA PHARMACEUTICAL 2014-12-31 CN disclosed
CN-104211618-A Process for producing pyrrole compound TAKEDA PHARMACEUTICAL 2014-12-17 CN disclosed
CN-102421753-A Process for preparing azole compounds TAKEDA PHARMACEUTICAL 2012-04-18 CN disclosed