SCHEMBL28816865

SCHEMBL28816865

Nc1cc(C(F)(F)F)cc(Cc2cccc(F)c2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
MPO P05164 3/20 0.46
NOS3 P29474 4/20 0.41
NOS1 P29475 4/20 0.41
NOS2 P35228 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
LTA4H P09960 1/20 0.40
BACE1 P56817 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
ADCY10 Q96PN6 1/20 0.39
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
IDO1 P14902 1/20 0.38
AGXT P21549 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28816893 0.79 NPC1 (0.50) NPC1RAB9AMPONOS3NOS1
SCHEMBL28000659 0.75 NPC1 (0.47) NPC1RAB9AMPONOS3NOS1
SCHEMBL28047019 0.73 ALDH1A1 (0.46) RAB9AMPONOS3NOS1NOS2
SCHEMBL29442814 0.71 L3MBTL1 (0.45) NPC1RAB9AMPONOS3NOS1
SCHEMBL21383967 0.71 L3MBTL1 (0.45) NPC1RAB9AMPONOS3NOS1
SCHEMBL28047795 0.69 L3MBTL1 (0.43) NPC1RAB9AMPOL3MBTL1TAAR1
SCHEMBL10569673 0.68 MPO (0.55) NPC1RAB9AMPONOS3NOS1
SCHEMBL562293 0.68 TACR1 (0.48) ADCY10
SCHEMBL5591246 0.68 ADCY10 (0.45) NPC1RAB9AMPOTAAR1ADCY10
SCHEMBL272886 0.68 NOS3 (0.54) RAB9ANOS3NOS1NOS2BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102482218-B Pyridine And Pyrazine Derivatives As Protein Kinase Modulators NOVARTIS AG 2015-01-21 CN disclosed