SCHEMBL288186

SCHEMBL288186

O=C1CCC(I)(C(=O)O)N1Cc1cccc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.46
LMNA P02545 2/20 0.46
PTGER4 P35408 4/20 0.46
S1PR1 P21453 1/20 0.46
GRK5 P34947 1/20 0.46
CDK8 P49336 1/20 0.46
S1PR5 Q9H228 1/20 0.46
PTGER2 P43116 1/20 0.45
ATM Q13315 1/20 0.45
KMT2A Q03164 2/20 0.44
NR4A2 P43354 1/20 0.44
FAAH O00519 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
MEN1 O00255 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
HTT P42858 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL290017 0.84 KMT2A (0.43) SMN1; SMN2PTGER4PTGER2KMT2ANR4A2
SCHEMBL4460381 0.82 HCRTR1 (0.41) KMT2AALDH1A1GAAMEN1
SCHEMBL288660 0.77 HTT (0.43) SMN1; SMN2LMNAPTGER4PTGER2KDM4E
SCHEMBL11099626 0.72 SMN1; SMN2 (0.58) SMN1; SMN2LMNAATMKDM4EALDH1A1
SCHEMBL289453 0.70 P2RX7 (0.60) SMN1; SMN2PTGER4S1PR1GRK5CDK8
SCHEMBL1611778 0.70 P2RX7 (0.60) SMN1; SMN2PTGER4S1PR1GRK5CDK8
SCHEMBL15967787 0.69 HSD11B1 (0.53) SMN1; SMN2LMNAS1PR1GRK5CDK8
SCHEMBL15967788 0.69 HSD11B1 (0.53) SMN1; SMN2LMNAS1PR1GRK5CDK8
SCHEMBL27723156 0.68 ATM (0.48) SMN1; SMN2LMNAPTGER4S1PR1GRK5
SCHEMBL4698249 0.67 KDM4E (0.70) SMN1; SMN2LMNAS1PR1GRK5CDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427429-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS Abbott GmbH & Co. KG (DE) 2012-03-14 EP disclosed
WO-2010128102-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS ABBOTT GMBH & CO. KG (DE) 2010-11-11 WO disclosed