SCHEMBL290017

SCHEMBL290017

O=C1CCC(I)(C(=O)O)N1Cc1cccc(F)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
PTGER4 P35408 1/20 0.43
PTGER2 P43116 1/20 0.43
HCAR2 Q8TDS4 1/20 0.41
NR4A2 P43354 1/20 0.41
FAAH O00519 1/20 0.41
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
CHRM5 P08912 2/20 0.40
KDM4E B2RXH2 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
FABP3 P05413 1/20 0.40
METAP2 P50579 1/20 0.40
FEN1 P39748 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM1 P11229 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL288660 0.85 HTT (0.43) PTGER4PTGER2ALDH1A1SMN1; SMN2KDM4E
SCHEMBL4460381 0.85 HCRTR1 (0.41) KMT2AMEN1ALDH1A1L3MBTL1
SCHEMBL288186 0.84 SMN1; SMN2 (0.46) KMT2AMEN1PTGER4PTGER2NR4A2
SCHEMBL288848 0.81 NPSR1 (0.57) KMT2AMEN1PTGER4PTGER2FAAH
SCHEMBL289516 0.81 FAAH (0.44) PTGER4FAAHALDH1A1L3MBTL1FEN1
SCHEMBL11888874 0.68 ALDH1A1 (0.56) KMT2AMEN1FAAHALDH1A1SMN1; SMN2
SCHEMBL288978 0.68 P2RX7 (0.55) KMT2AMEN1ALDH1A1SIGMAR1
SCHEMBL1611845 0.68 P2RX7 (0.55) KMT2AMEN1ALDH1A1SIGMAR1
SCHEMBL30601818 0.67 MEN1 (0.46) KMT2AMEN1HCAR2NR4A2ALDH1A1
SCHEMBL26123725 0.67 MEN1 (0.46) KMT2AMEN1HCAR2NR4A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427429-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS Abbott GmbH & Co. KG (DE) 2012-03-14 EP disclosed
WO-2010128102-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS ABBOTT GMBH & CO. KG (DE) 2010-11-11 WO disclosed