SCHEMBL28819152

SCHEMBL28819152

NC(=O)c1cccc(C(F)(F)F)c1C1CCCC1N1CCCC1

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.41
PARP1 P09874 1/20 0.39
PNMT P11086 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28819153 1.00 HTR1A (0.41) HTR1APARP1PNMT
SCHEMBL28015407 0.90 HTR1A (0.36) HTR1A
SCHEMBL28014792 0.79 SLC6A9 (0.40)
SCHEMBL28014793 0.79 SLC6A9 (0.40)
SCHEMBL7793147 0.77 AKR1C3 (0.41)
SCHEMBL4181858 0.77 PNMT (0.43) PARP1PNMT
Hydrochloric Acid SCHEMBL7798727 0.76 AKR1C3 (0.40)
SCHEMBL28093498 0.76 TAS1R3 (0.45) PARP1PNMT
SCHEMBL1514836 0.74 HSD11B1 (0.48) PARP1
SCHEMBL1514789 0.74 NOS3 (0.41) PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102482203-B Carbocyclic GLYT1 receptor antagonists HOFFMANN LA ROCHE 2015-06-03 CN disclosed