SCHEMBL28832869

SCHEMBL28832869

O=COC(Cc1cn[nH]c1)Cc1ccccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 1/20 0.38
PTPRA P18433 1/20 0.38
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
GRIN3A Q8TCU5 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
NAMPT P43490 3/20 0.34
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
PGR P06401 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
PTGS1 P23219 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27808924 0.77 ROCK2 (0.36) ROCK2ROCK1
SCHEMBL27545407 0.77 FFAR1 (0.38)
SCHEMBL28047241 0.76 NOS2 (0.33) ROCK2
SCHEMBL28787513 0.76 ROCK1 (0.37) NAMPTROCK2ROCK1
SCHEMBL27972554 0.76 ROCK2 (0.41) NAMPTROCK2SLC6A4
SCHEMBL27809130 0.75 ALDH1A1 (0.35) SMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL27525176 0.75 NOS2 (0.40) NAMPT
SCHEMBL28824812 0.74 ALDH1A1 (0.36) KDM4EALDH1A1MAPTTSHR
SCHEMBL28868753 0.74 LDHA (0.41) SMN1; SMN2ALDH1A1NAMPTROCK2ROCK1
SCHEMBL23075459 0.73 L3MBTL1 (0.50) SMN1; SMN2ALDH1A1CYP1A2CYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105849096-B Piperidine derivatives having multimodal activity against pain 埃斯蒂文制药股份有限公司 2019-11-29 CN disclosed
CN-105849096-A Piperidine derivatives having multimodal activity against pain 埃斯蒂文博士实验室股份有限公司 2016-08-10 CN disclosed