SCHEMBL28868753

SCHEMBL28868753

COc1ccc(CC(Cc2cn[nH]c2)OC=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.41
NAMPT P43490 1/20 0.40
SLC6A4 P31645 1/20 0.40
ROCK2 O75116 2/20 0.39
ROCK1 Q13464 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
ACACB O00763 1/20 0.37
PLCG1 P19174 1/20 0.36
PTGDR Q13258 1/20 0.35
NOS2 P35228 1/20 0.35
POLB P06746 1/20 0.35
GFER P55789 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
ALOX12 P18054 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27545407 0.84 FFAR1 (0.38) ACACB
SCHEMBL28787513 0.83 ROCK1 (0.37) NAMPTROCK2ROCK1ACACBNOS2
SCHEMBL28047241 0.83 NOS2 (0.33) ROCK2ACACBNOS2
SCHEMBL27972554 0.83 ROCK2 (0.41) NAMPTSLC6A4ROCK2NOS2
SCHEMBL27525176 0.80 NOS2 (0.40) NAMPTNOS2
SCHEMBL28858540 0.78 NOS2 (0.36) NOS2
SCHEMBL28825902 0.77 LDHA (0.40) LDHASLC6A4CYP1A2CYP2D6CYP2C19
SCHEMBL27809130 0.77 ALDH1A1 (0.35) ALDH1A1SMN1; SMN2
SCHEMBL28816888 0.75 CTSK (0.36) NOS2
SCHEMBL28790153 0.74 LDHA (0.35) LDHASLC6A4POLBALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109071546-A Pyrazolo [1,5-A ] pyrazin-4-yl derivatives as JAK inhibitors 辉瑞大药厂 2018-12-21 CN disclosed