SCHEMBL28047241

SCHEMBL28047241

O=COC(Cc1ccc(CCl)cc1)Cc1cn[nH]c1

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 1/20 0.33
ACACB O00763 1/20 0.32
ROCK2 O75116 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27972554 0.89 ROCK2 (0.41) NOS2ROCK2
SCHEMBL28787513 0.86 ROCK1 (0.37) NOS2ACACBROCK2
SCHEMBL28868753 0.83 LDHA (0.41) NOS2ACACBROCK2
SCHEMBL27809130 0.82 ALDH1A1 (0.35)
SCHEMBL27545407 0.81 FFAR1 (0.38) ACACB
SCHEMBL27525176 0.79 NOS2 (0.40) NOS2
SCHEMBL28047249 0.78 KLKB1 (0.37) ROCK2
SCHEMBL28832869 0.76 FDPS (0.38) ROCK2
SCHEMBL27808924 0.76 ROCK2 (0.36) NOS2ROCK2
SCHEMBL28052289 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143201-B Benzyl amine derivative 卡尔维斯塔制药有限公司 2019-02-22 CN disclosed
CN-105143201-A Benzylamine derivatives KALVISTA PHARMACEUTICALS LTD 2015-12-09 CN disclosed