SCHEMBL28900568

SCHEMBL28900568

O=C(c1ccc(N2CCOCC2)cc1)N1CC[CH]CC1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.59
HSD11B1 P28845 1/20 0.58
ALDH1A1 P00352 4/20 0.57
KDM4E B2RXH2 3/20 0.57
MAPT P10636 1/20 0.57
HTT P42858 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
PHGDH O43175 1/20 0.57
ALOX15 P16050 1/20 0.54
HSD17B10 Q99714 1/20 0.54
GSK3B P49841 1/20 0.54
AKR1C3 P42330 1/20 0.51
TP53 P04637 1/20 0.51
KMT2A Q03164 1/20 0.51
MAPK1 P28482 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
MGLL Q99685 1/20 0.50
TSHR P16473 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14528664 0.82 HPGD (0.65) HPGDHSD11B1ALDH1A1KDM4EMAPT
SCHEMBL10720943 0.80 PHGDH (0.81) HPGDALDH1A1KDM4EMAPTHTT
SCHEMBL4618652 0.80 ALDH1A1 (0.84) HPGDALDH1A1KDM4EMAPTHTT
SCHEMBL1359639 0.79 HPGD (0.63) HPGDHSD11B1ALDH1A1KDM4EMAPT
SCHEMBL22387605 0.78 HSD11B1 (0.62) HPGDHSD11B1ALDH1A1KDM4EMAPT
SCHEMBL2742813 0.77 NPC1 (0.66) HPGDALDH1A1KDM4EMAPTHTT
SCHEMBL3824666 0.77 GSK3B (0.66) HPGDALDH1A1KDM4EMAPTHTT
SCHEMBL7403944 0.75 HPGD (0.55) HPGDALDH1A1MAPTHTTPHGDH
SCHEMBL60648 0.75 KMO (0.67) HPGDALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL28296651 0.75 HPGD (0.86) HPGDALDH1A1KDM4EMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112370452-A Heterocyclic amides as kinase inhibitors 葛兰素史密斯克莱知识产权发展有限公司 2021-02-19 CN disclosed
CN-107624111-B Heterocyclic amides as kinase inhibitors 葛兰素史密斯克莱知识产权发展有限公司 2020-11-03 CN disclosed