SCHEMBL28908256

SCHEMBL28908256

OB(O)c1csc(COc2ccccc2F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.41
DAO P14920 1/20 0.39
LMNA P02545 1/20 0.37
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
LIPE Q05469 1/20 0.36
FKBP1A P62942 1/20 0.35
MAPT P10636 3/20 0.34
KDM5A P29375 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28519499 0.83 RXRA (0.40) ALDH1A1L3MBTL1TDP1LIPEMAPT
SCHEMBL28521420 0.83 ALDH1A1 (0.45) MRGPRX4LMNAALDH1A1L3MBTL1LIPE
SCHEMBL28521446 0.80 NPC1 (0.39) ALDH1A1L3MBTL1TDP1KMT2AFFAR1
SCHEMBL28512482 0.79 ENPP2 (0.42) DAOL3MBTL1MAPTENPP2
SCHEMBL28520513 0.79 CA1 (0.41) DAOLMNAALDH1A1L3MBTL1HDAC6
SCHEMBL28520033 0.77 MAOB (0.41) MRGPRX4DAOLMNAHDAC1HDAC6
SCHEMBL15332082 0.74 LMNA (0.43) MRGPRX4DAOLMNAALDH1A1L3MBTL1
SCHEMBL28520517 0.71 ACHE (0.44) LMNAALDH1A1L3MBTL1TDP1MAPT
SCHEMBL28529096 0.71 NPC1 (0.42) ALDH1A1L3MBTL1MAPTMEN1KMT2A
SCHEMBL28521411 0.70 ENPP2 (0.51) MRGPRX4LMNAALDH1A1ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602834-B Bruton's tyrosine kinase inhibitor 北京盛诺基医药科技股份有限公司 2021-01-08 CN disclosed