SCHEMBL28972700

SCHEMBL28972700

C/C(=C\c1cc(-c2ccc(C#N)c(Cl)c2)cs1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EIF4E P06730 3/20 0.42
ABL1 P00519 1/20 0.41
CASP1 P29466 1/20 0.39
CYP11B2 P19099 4/20 0.39
SLC22A12 Q96S37 2/20 0.39
CYP11B1 P15538 2/20 0.37
NR3C2 P08235 1/20 0.36
AR P10275 3/20 0.35
S1PR1 P21453 1/20 0.35
S1PR5 Q9H228 1/20 0.35
S1PR3 Q99500 1/20 0.35
TRPV4 Q9HBA0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28972450 0.90 CASP1 (0.43) EIF4EABL1CASP1CYP11B2SLC22A12
SCHEMBL28972699 0.85 CYP11B2 (0.48) CYP11B2SLC22A12CYP11B1
SCHEMBL28972684 0.82 RXRA (0.52) AR
SCHEMBL28972437 0.81 MAPT (0.41) EIF4ECASP1CYP11B2SLC22A12NR3C2
SCHEMBL28972415 0.80 MMP3 (0.39)
SCHEMBL30112097 0.80 CYP11B2 (0.46) EIF4EABL1CASP1CYP11B2SLC22A12
SCHEMBL28972451 0.77 RORC (0.46) EIF4ECYP11B2SLC22A12CYP11B1AR
SCHEMBL28972703 0.76 CYP11B2 (0.46) CYP11B2CYP11B1
SCHEMBL379474 0.75 AKR1C3 (0.50)
SCHEMBL379475 0.75 AKR1C3 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110016011-B Amide derivative and medical use thereof 北京美倍他药物研究有限公司 2023-02-03 CN disclosed