SCHEMBL29024488

SCHEMBL29024488

CC(C)COc1ccc(Cn2nc(C3CCNCC3)cc2CC2CC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.39
HTR2A P28223 7/20 0.36
SLC16A3 O15427 2/20 0.34
SLC16A1 P53985 2/20 0.34
MCTS1 Q9ULC4 2/20 0.34
PDE6D O43924 1/20 0.33
PRMT5 O14744 1/20 0.33
GCGR P47871 1/20 0.33
GIPR P48546 1/20 0.33
ALK Q9UM73 1/20 0.33
GPR4 P46093 1/20 0.33
IKBKB O14920 1/20 0.32
FAAH O00519 1/20 0.32
KCNH2 Q12809 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29024482 0.88 HTR2A (0.40) ABL1HTR2AKCNH2HTR2C
SCHEMBL29024487 0.87 HRH1 (0.40) ABL1HTR2ASLC16A3SLC16A1MCTS1
SCHEMBL29024489 0.83 ABL1 (0.39) ABL1HTR2ASLC16A3SLC16A1MCTS1
SCHEMBL30478116 0.80 LMNA (0.36) HTR2ASLC16A3SLC16A1MCTS1FAAH
SCHEMBL30478103 0.77 LTA4H (0.36) FAAH
SCHEMBL29024635 0.77 TP53 (0.39) HTR2APRMT5FAAH
SCHEMBL29024637 0.76 HTR2A (0.47) HTR2AKCNH2HTR2C
SCHEMBL29024639 0.74 SLC16A3 (0.41) ABL1HTR2ASLC16A3SLC16A1MCTS1
SCHEMBL29024481 0.71 HTR2A (0.42) ABL1HTR2AKCNH2HTR2C
SCHEMBL30478119 0.69 SLC16A3 (0.38) SLC16A3SLC16A1MCTS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116354925-A Pyrazole derivatives and use thereof 江苏恩华药业股份有限公司 2023-06-30 CN claimed
CN-116354925-A Pyrazole derivatives and use thereof 江苏恩华药业股份有限公司 2023-06-30 CN disclosed