SCHEMBL2902878

SCHEMBL2902878

N#Cc1ccc(Oc2nc[c]cc2Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
CYP2C9 P11712 2/20 0.40
TSHR P16473 1/20 0.40
APEX1 P27695 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MAPK1 P28482 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP19A1 P11511 1/20 0.40
MERTK Q12866 1/20 0.39
PARP15 Q460N3 1/20 0.37
PARP10 Q53GL7 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
MEN1 O00255 2/20 0.36
RAB9A P51151 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
IL18 Q14116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2897638 0.83 CYP2C9 (0.49) LMNACYP2C9TSHRAPEX1SMN1; SMN2
SCHEMBL6629345 0.80 PIN1 (0.43) LMNACYP2C9TSHRAPEX1SMN1; SMN2
SCHEMBL2897637 0.77 LMNA (0.39) LMNACYP2C9TSHRAPEX1SMN1; SMN2
SCHEMBL2903002 0.77 SMN1; SMN2 (0.42) LMNACYP2C9TSHRAPEX1SMN1; SMN2
SCHEMBL30689412 0.76 CYP19A1 (0.51) LMNACYP2C9TSHRAPEX1SMN1; SMN2
SCHEMBL10355081 0.75 MERTK (0.43) LMNAMAPK1CYP19A1MERTKPARP15
SCHEMBL2900255 0.75 PTGS2 (0.39) LMNACYP2C9TSHRAPEX1SMN1; SMN2
SCHEMBL2901895 0.75 HSPB1 (0.44) LMNASMN1; SMN2MAPK1L3MBTL1MERTK
SCHEMBL6581279 0.73 F10 (0.53) LMNACYP2C9TSHRAPEX1SMN1; SMN2
SCHEMBL11377102 0.72 CYP19A1 (0.46) LMNACYP2C9SMN1; SMN2MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100305124-A1 Acylated Aminopyridine and Aminopyridazine Insecticides BAYER CROPSCIENCE AG (DE) 2010-12-02 US disclosed
EP-2236505-A1 Acylated aminopyridines and pyridazines as insecticides Bayer CropScience AG (DE) 2010-10-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100305124-A1 Acylated Aminopyridine and Aminopyridazine Insecticides AAAS, DDT, QDPR LMNA 2262/4885CYP2C9 310/4885TSHR 2740/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.