SCHEMBL29201807

SCHEMBL29201807

CC(=O)c1cc(C)c(C(=O)NCC(=O)NC(F)C(F)F)s1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR139 Q6DWJ6 6/20 0.32
SLC6A9 P48067 4/20 0.32
PPARG P37231 1/20 0.32
NR2E3 Q9Y5X4 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
SLC6A5 Q9Y345 2/20 0.31
ALOX15 P16050 1/20 0.31
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
USP5 P45974 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
PSMB11 A5LHX3 1/20 0.30
PSMA7 O14818 1/20 0.30
PSMB1 P20618 1/20 0.30
PSMA1 P25786 1/20 0.30
PSMA2 P25787 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19457471 0.79 LMNA (0.43) KDM4EALDH1A1HPGDPOLBKMT2A
SCHEMBL29181724 0.77 GPR139 (0.32) GPR139KMT2A
SCHEMBL29098708 0.73 SLC6A9 (0.39) GPR139SLC6A9ALDH1A1HPGDSLC6A5
SCHEMBL24993293 0.70 KDM4E (0.45) KDM4EALDH1A1HPGDPOLBKMT2A
SCHEMBL29012853 0.67 GPR139 (0.42) GPR139SLC6A9PPARGNR2E3NCOR2
SCHEMBL28863527 0.67 SLC6A9 (0.35) GPR139SLC6A9ALDH1A1HPGDSLC6A5
SCHEMBL16334956 0.65 DAO (0.50) KDM4EALDH1A1ALOX15KMT2A
SCHEMBL13994843 0.64 ALOX15 (0.44) KDM4EALDH1A1HPGDALOX15KMT2A
SCHEMBL29201822 0.63 DAO (0.41) KDM4EALDH1A1HPGDALOX15POLB
SCHEMBL28863530 0.62 EGLN1 (0.35) GPR139ALDH1A1KMT2ATDP1PSMB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117447443-A Method for preparing rotirana intermediate by one-pot method 北京康立生医药技术开发有限公司 2024-01-26 CN claimed
CN-117447443-A Method for preparing rotirana intermediate by one-pot method 北京康立生医药技术开发有限公司 2024-01-26 CN disclosed