SCHEMBL29314126

SCHEMBL29314126

CCN(c1ccc(F)c(C)n1)C(O)Cc1c(-c2cn[nH]c2)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 11/20 0.34
ROCK1 Q13464 11/20 0.34
MTOR P42345 1/20 0.31
PIK3CA P42336 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29314121 0.70 POLQ (0.44) ROCK2ROCK1
SCHEMBL29315913 0.66 ROCK1 (0.39) ROCK2ROCK1
SCHEMBL29315909 0.66 ROCK2 (0.46) ROCK2ROCK1
SCHEMBL29316278 0.64 NPBWR1 (0.39) ROCK2ROCK1
SCHEMBL29316276 0.58 ROCK2 (0.39) ROCK2ROCK1
SCHEMBL31009157 0.57 POLQ (0.46) ROCK2ROCK1
SCHEMBL13036088 0.56 LRRK2 (0.50) ROCK2ROCK1
SCHEMBL25795129 0.55 NOTUM (0.46) ROCK1
SCHEMBL20040983 0.55 NPBWR1 (0.44) ROCK2ROCK1
SCHEMBL28199128 0.55 ROCK2 (0.44) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed