SCHEMBL29316276

SCHEMBL29316276

FC(F)(F)c1cc(-c2cn[nH]c2)c(OCc2ccccc2)c(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.39
ROCK1 Q13464 3/20 0.39
PRMT5 O14744 1/20 0.39
METAP2 P50579 1/20 0.38
PTPN2 P17706 2/20 0.38
PTPN1 P18031 2/20 0.38
PTPN6 P29350 2/20 0.38
GRK2 P25098 2/20 0.38
RXRA P19793 2/20 0.37
RXRB P28702 2/20 0.37
RXRG P48443 2/20 0.37
AKT1 P31749 1/20 0.37
AKT2 P31751 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 1/20 0.37
PTGER1 P34995 2/20 0.37
CYP2C9 P11712 1/20 0.37
FEN1 P39748 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15898915 0.73 RXRA (0.42) PTPN2PTPN1PTPN6RXRARXRB
SCHEMBL29316278 0.72 NPBWR1 (0.39) ROCK2ROCK1METAP2PDK2
SCHEMBL29315913 0.70 ROCK1 (0.39) ROCK2ROCK1RXRARXRBRXRG
SCHEMBL29317047 0.70 HTT (0.44) PTPN2PTPN1PTPN6RXRARXRB
SCHEMBL17276683 0.69 TRPA1 (0.55) ROCK2ROCK1AKT1AKT2FEN1
SCHEMBL24896625 0.68 AKT1 (0.42) ROCK2ROCK1PRMT5GRK2AKT1
SCHEMBL30847795 0.68 CYP1A2 (0.41) PTPN2PTPN1PTPN6RXRARXRB
SCHEMBL19920979 0.66 PIN1 (0.47) ROCK2AKT1AKT2MEN1ALDH1A1
SCHEMBL6257616 0.66 AKT2 (0.59) ROCK2PRMT5AKT1AKT2MEN1
SCHEMBL4051954 0.65 AKT1 (0.54) ROCK2PRMT5GRK2AKT1AKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed