SCHEMBL29314449

SCHEMBL29314449

CNc1ncc(C#N)c(NCC2CCCN2)n1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.49
MAP3K8 P41279 1/20 0.46
MERTK Q12866 3/20 0.44
PRKCQ Q04759 5/20 0.44
SYK P43405 3/20 0.43
KCNH2 Q12809 3/20 0.43
MAPK3 P27361 1/20 0.43
MAPK1 P28482 1/20 0.43
AURKB Q96GD4 1/20 0.43
EHMT2 Q96KQ7 1/20 0.39
LRRK2 Q5S007 2/20 0.38
BCDIN3D Q7Z5W3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29313569 0.78 TNK2 (0.48) CHEK1MAP3K8MAPK1
SCHEMBL29313579 0.76 KAT2B (0.42) MAP3K8PRKCQLRRK2
SCHEMBL29313573 0.74 LRRK2 (0.47) CHEK1PRKCQLRRK2
SCHEMBL23019347 0.71 PRKCQ (0.41) PRKCQSYKLRRK2
SCHEMBL29313773 0.71 CCNA2 (0.46) MERTKPRKCQSYKLRRK2
SCHEMBL1598417 0.70 CHEK1 (0.46) CHEK1MAP3K8
SCHEMBL1598420 0.70 CHEK1 (0.46) CHEK1MAP3K8
SCHEMBL29313719 0.69 AURKA (0.38) SYKLRRK2
SCHEMBL29313606 0.69 PTK2 (0.40) PRKCQSYKLRRK2
SCHEMBL1598410 0.68 MAP3K8 (0.42) CHEK1MAP3K8SYKKCNH2EHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed