SCHEMBL30847795

SCHEMBL30847795

FC(F)(F)c1cc(N2CCCC2)c(OCc2ccccc2)c(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KCNQ2 O43526 1/20 0.40
SLC6A4 P31645 4/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HTR1A P08908 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A3 Q01959 1/20 0.39
RPS6KB1 P23443 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30847650 0.79 ALOX5 (0.39) SLC6A4ALDH1A1MEN1KMT2AHTR1A
SCHEMBL15898915 0.76 RXRA (0.42) SLC6A4ALDH1A1MEN1KMT2AHTR2C
SCHEMBL30847726 0.75 DRD2 (0.38) ALDH1A1MEN1KMT2APTPN2PTPN1
SCHEMBL30847657 0.75 SCN5A (0.43) PTPN2PTPN1PTPN6RXRARXRB
SCHEMBL29317047 0.75 HTT (0.44) HTTSLC6A4ALDH1A1MEN1KMT2A
SCHEMBL30847704 0.73 AR (0.36) SLC6A4ALDH1A1MEN1KMT2ARPS6KB1
SCHEMBL30847744 0.73 AR (0.36) SLC6A4ALDH1A1MEN1KMT2ARPS6KB1
SCHEMBL17048680 0.73 SIGMAR1 (0.45) RXRARXRBRXRGHRH3LTA4H
SCHEMBL12774184 0.69 HTR1A (0.36) CYP1A2CYP2D6MAPTCYP2C19SMN1; SMN2
SCHEMBL16046661 0.68 HTR1A (0.74) MAPTSMN1; SMN2NPSR1SLC6A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4598901-A1 PYRROLIDINE AND IMIDAZOLIDINE BASED DNA POLYMERASE THETA INHIBITORS AND USE THEREOF Thomas Jefferson University (US) 2025-08-13 EP disclosed
WO-2024076964-A1 PYRROLIDINE AND IMIDAZOLIDINE BASED DNA POLYMERASE THETA INHIBITORS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-04-11 WO disclosed